Hauora, Mau faaineineraa
Raau "Velaksin": mua manawanui, tohutohu mo te whakamahi, analogs
Ka taea e te hoko e ahau pōuritanga kahore te whakahaunga? E kore te mea nui te rārangi o taua hua. Ko e tika ana ki te meka e taea e ratou faatîtîraa, me te ope o ngā pānga taha tenei. Na reira, i mua i te tango i taua tikanga, kia mohio ki te haere ki te tohunga.
mōhiohio whānui
e kore te Depression tukinotia e te raau taero. Otiia ki te whakapai ake i te mahi o te pūnaha io, whakahau tonu maha kaiwhakaako ki o ratou tūroro ngā pōuritanga. Ko tētahi o ratou ko te tarukino "Velaksin". Ka kia te aroaro o Mua e pā ana ki tenei taputapu me ona āhuatanga, me ngā tohutohu mō te whakamahi i raro.
Ko te hanganga o te raau taero, tona ahua o production
I roto i te aha puka hua reira he raau rite "Velaksin"? Papa me capsules - he anake nga momo o te tarukino.
He ma Papa "Velaksin", i whaoa nei ki tetahi taha "E741", me te āhua flat porohita me te chamfer. Ratou whakauru kaha he venlafaxine, māngai nei i roto i te puka o te hydrochloride. whakaurua hoki i roto i tenei rongoā ngā wāhanga ngaahi houalotú pērā i anhydrous colloidal takawai, monohydrate reihuka, te konutai māngaro glycolate, stearate konupora me te MCC.
papa Kikī i roto i mōkihi namunamu me kātene aua.
Drug "Velaksin" - capsules, tohutohu hoki te whakamahi i E kopakia ana i roto i te tākai, pepa, gelatin me te mārō. E ratou pōtae karaka-parauri, me te tïpako taekore. Ko hoki te wāhanga kaha o tenei puka te venlafaxine pūhui. I tua atu ki tona hanganga o tenei rongoā ngā kai atu.
Ka rite ki nga mahi tarukino?
"Velaksin" - he whakatupuranga hou o anti-depressant. E ai ki te hanganga matū o tona taonga kaha e kore e no ki tetahi piha mohiotia o pōuritanga (hei tauira, tricyclic, tetracyclic, atu ranei). Tohunga mea e te tarukino he kaha enantiomer 2 racemate.
pā ana te parau tumu o te mahi o tenei tarukino te ki tona kaha ki te potentiate te CNS karere hihiko te tuku.
E ai ki nga tohutohu, venlafaxine me tona metabolite matua (EFA ranei e-desmetilvenlafaksin) tohu inhibitors puai o te reuptake o norepinephrine me serotonin me inhibitors ngoikore o te dopamine reuptake. E kore e taea e tatou te mea e, teie mau matū e taea ki te whakaiti i te mahi beta-adrenergic i muri i te rongoā kotahi, me te tamau. He rite whai hua ki reuptake o neurotransmitters EFA me venlafaxine.
He aha atu he tarukino faahiahia "Velaksin"? pūrongo Guide e te whakauru kaha o te tarukino he hunaonga ki a te mau farii ohipa N- me m-cholinergic, roro α1-adrenoceptors me histamine H1-receptors. I tua atu, inhibits reira te mahi o Mao me e kore faitatau ki fentsiklidinovymi, opioid, benzodiazepine me NMDA-receptors.
Ko te kinetics o te tarukino
ahakoa horomia te tarukino te, "Velaksin" (papa)? kī Tohutohu mō te Whakamahi e te tino pai whenumi te wāhanga hohe o tenei tarukino i te punuatuna. I muri i te horopeta kotahi o te medicament i roto i te inenga o 25-150 mg o tona kukū rawa i roto i te toto tae te i muri i 2.4 haora. Ko te kupu venlafaxine te ngā metabolized i roto i te haere tuatahi i roto i te ate. Ki te tangohia te tarukino i te kai, i te ona kukū piki tihi e 27-30 meneti i roto i te wē.
whakaaro te metabolite matua te he te tikanga o te e-desmetilvenlafaksin. Ko tōna hawhe-te ora me te whakakorenga hawhe-ora o te venlafaxine he 11 me te 5 haora, aua (putanga i roto i te puka tonu i nga whatukuhu).
Ko te kinetics o raau taero i roto i te āhuatanga haumanu motuhake
hiahiatia Drug "Velaksin" ako te pānui i roto i te iwi ki te cirrhosis o te ate he atu āhuatanga nekeneke. toto kukū o te raau taero nui haere i roto i enei tūroro, me tona tere o te papī, i runga i te anga ke, iti.
I roto i te kino iti hoki tākihi, täkihi me te āhua whakawātea katoa iti EFA me venlafaxine te ka roa te whakakorenga wā hawhe-ora te.
Me mahara hoki käore te reira e kore e te ira tangata me te tau o te manawanui pā te pharmacokinetics o te tarukino i raro i whakaarohia.
Tuhinga hoki
Aha tatou e hinaaro ai i te taputapu pērā i "Velaksin"? Ko te whakamahi o tenei tarukino whakaaturia i roto i te whārua o ngā takenga (mo te maimoatanga me te prophylaxis).
Ūhia ki te whakarite
I raro i te mea e kore e taea e tikanga te whakamahi i te tarukino "Velaksin"? Reviews o tūroro me kaiwhakaako titau e contraindicated tenei tarukino te ki riro:
- i te fariiraa i Mao inhibitors ;
- i roto i disorders tākihi nui;
- i roto i te hapū whakapae whakapumautia ranei;
- i roto i disorders nui o te ate;
- i roto i te whāngai ū;
- i roto i te taiohitanga me tamarikitanga, e ko, tae noa ki te tau o te nuinga;
- ki te tūtohutanga tiketike ki te tarukino.
I tua atu, kia āta tangohia tenei tarukino i roto i angina iu, nui haere infarction myocardial (tae atu i te hou heke), takawhita, hītori haehae, tachycardia, mate taimaha, pēhanga intraocular, koki-katinga papahewa, predisposition ki toto i mucous me kiri, āhua härukiruki.
Drug "Velaksin" (papa): tohutohu mō te whakamahi
Raau "Velaksin" anake kia tangohia i roto i te kai. Ko te horopeta tīmatanga tūtohutia o te tarukino ko 75 mg, wehea i roto i te 2 werohanga wehea (i.e., 37.5 mg rua he ra), i tenei ra.
Ki te i muri i te maha o ngā wiki o therapy, e kore kua huru o te manawanui ake, kua nui haere te horopeta rā ki te 150 mg te ra, i roto i rua pota wehea (i.e., 75 mg rua he ra).
Ki te titau te manawanui he horopeta teitei o te raau (hei tauira, nui whakararuraru fakalotofo'í, ranei te tahi atu tikanga tono therapy pahoho), ka taea te kaitoi tautapa 150 mg o tarukino i roto i te 2 haora, a ka āta whakanui i te horopeta e 75 mg (2-3 ra i muri mai) ki te whakatutuki i te hua e hiahiatia ana.
E ai ki nga tohutohu, te inenga mōrahi "Velaksina" ko 375 mg ia ra. I muri te whakatutuki i te pānga e hiahiatia, e taea te āta tuku iho reira ki te taumata iti.
ārai matahoki me te tiaki therapy
tiaki tautoko o nga moni e taea te tango i te ono marama. I roto i tenei take, te rongoā tangohia i roto i te pota iti.
I roto i te iti hoki tākihi ngawari hiahiatia ako dosing talena te. I roto i te mate rite tūtohutia raro horopeta āhua i te 25-50%. Me mahara hoki käore te reira e kore e tika kia whakamahia venlafaxine i roto i nui iti hoki tākihi, mai kore ngā mōhiohio i runga i te haumaru o taua therapy ki te rā, e kore.
Iwi e te hunga i runga i tātari toto, kia riro 50% o te inenga mua rā o te raau taero i muri i nga pito wātū.
Hoki ngawari iti hoki te ako dosing talena ate kore hoki te hiahiatia. A, no te te mate, ko te kia heke horopeta āhua i te 50%. Ki te whakaaro ki kino kore ate, i roto i tenei take rāhuitia te whakamahi o te venlafaxine te.
I roto i te paari, kia whakamahia te tarukino "Velaksin" ki te tūpato tino. Ko e tika ana ki te tūkino taea o nga whatukuhu tenei. Me whakahau te tūroro i te horopeta whai hua i raro. I roto i tenei take, kia waiho te manawanui i raro i te tirotiro tamau hauora.
Whakakore raau
Runga ki te whakaotinga o te fariiraa i te tarukino kia whakaaro ki te whakaiti i te horopeta āta (i roto i te wiki). Kei te hiahiatia te reira ki te mau i te huru o te manawanui, i roto i te tikanga ki te whakaiti i te tūponotanga o tauhohe kino e pā ana ki te whakakāhoretanga o te tarukino.
Ko te wa e hiahiatia ana mo te mutunga oti o te rongoā, tei runga i te inenga, roanga o te therapy me takitahi ki takitahi.
pānga taha
He aha e nga pānga e hiahiatia o te tarukino e taea meinga "Velaksin"? Mua mea e te whanaketanga o te hunga ranei era atu meatanga kino e whai ake nei i te whakamahi o tenei taputapu, tei runga i te horopeta riro.
Ko te tauhohe tino auau te whakakitenga mai āhua tōraro ngā te whai ake:
- takawhita, heke hiahia, moe rerekē, kōroke, ohoroa, whakapairuaki, Makere o, tremors, ruaki, cramps uaua, mangai maroke te kiri;
- moemoea, kakā, mate taimaha, tachycardia, hyponatremia, tau'a, hypotension postural, whanoke, tauhohenga härukiruki, excitability manavasii, puare noa, paresthesia, syndrome neuroleptic, hiamoe, syndrome serotonergic;
- nui haere oro uaua, hukihuki, dysuria, photosensitivity, te pupuri mimi, anorgasmia;
- toto i roto i te kiri, ejaculation rerekē, menorrhagia, heke libido, sweating;
- thrombocytopenia, raruraru noho, erythema multiforme, mydriasis, Stevens - Johnson, raruraru ataata, reka waimaero, Tuhinga o wa, ngoikore, ponana kiri, rohirohi, toto tauhohe anaphylactic.
tūtohutanga
Hokona ahakoa pōuritanga kahore te whakahaunga? e kore he tino nui te rārangi o enei rongoa ( "Prozac", "Paxil", "Despres", "Azafen", "Pahi", "amitriptyline"), me te tarukino "Velaksin" Kei te kore ngā i roto i reira. E hoko i te reira i roto i pharmacies, taea e koe anake i te whakahaunga o te tākuta.
I mua i te tango i tēnei rongoā i raro i te arotake, rawa tūroro ki disorders fakalotofo'í, kia whakaaro te tūponotanga nui o ngā nganatanga suicidal. I roto i tenei whakaaro, i te timatanga o te therapy tarukino tūtohutia hoki te whakamahi i roto i te horopeta iti me i raro i tata te tirotiro hauora.
Iwi ki disorders huru i roto i te maimoatanga ki pōuritanga kia whakawhanake āhua härukiruki hypomanic ranei.
kia tino ki te whakatupato o te hiahia ki te kite i tonu he tākuta i te take o ngā huānga urticaria, rashes mate pāwera ranei tūroro.
Ētahi tūroro i roto i te tukanga o te fariiraa i venlafaxine kitea he hua horopeta-ti'aturi i roto i te pēhanga toto.
kia whakatupato tūroro ruhiruhia o te ofatiraa taea o te tikanga o te pauna, me te whanoke whanaketanga.
I roto i te maimoatanga o te moni kia karo tango inu waipiro.
Raau "Velaksin": mua manawanui, analogues hua
He aha te iwi e mea e pā ana ki tenei tarukino ki te manawanui? Kua korerotia maha kiritaki he maha nui o ngā pānga taha e puta i te tango i tēnei rongoā. Tino maha tenei tarukino ai tauhohe kino pērā i te momoe, ngoikore, ohoroa, hukihuki, whakaaro rerekē, whārua me te whakama. I tua atu, titau te tahi mau tūroro e noho enei pānga i muri i te otinga o te maimoatanga. Ano, he maha ngā kaiwhakamahi amuamu e pā ana ki te ahua o tohu withdrawal , me te ti'aturiraa.
He aha e taea e whakakapi raau pērā i "Velaksin"? Kei te kore ki te e kitea Analogs o tenei tarukino i roto i drugstores katoa. Ka rite ki te tikanga, ngā tohunga enei te whai ake: "Venlafaxine Sandoz", "Efevelon", "Alvent", "Nyuvelong", "Velafaks", "Dapfiks", "Voksemel", "Venlaksor", "Vensuert", "venlafaxine".
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