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Raau "Velaksin": mua manawanui, tohutohu mo te whakamahi, analogs

Ka taea e te hoko e ahau pōuritanga kahore te whakahaunga? E kore te mea nui te rārangi o taua hua. Ko e tika ana ki te meka e taea e ratou faatîtîraa, me te ope o ngā pānga taha tenei. Na reira, i mua i te tango i taua tikanga, kia mohio ki te haere ki te tohunga.

mōhiohio whānui

e kore te Depression tukinotia e te raau taero. Otiia ki te whakapai ake i te mahi o te pūnaha io, whakahau tonu maha kaiwhakaako ki o ratou tūroro ngā pōuritanga. Ko tētahi o ratou ko te tarukino "Velaksin". Ka kia te aroaro o Mua e pā ana ki tenei taputapu me ona āhuatanga, me ngā tohutohu mō te whakamahi i raro.

Ko te hanganga o te raau taero, tona ahua o production

I roto i te aha puka hua reira he raau rite "Velaksin"? Papa me capsules - he anake nga momo o te tarukino.

He ma Papa "Velaksin", i whaoa nei ki tetahi taha "E741", me te āhua flat porohita me te chamfer. Ratou whakauru kaha he venlafaxine, māngai nei i roto i te puka o te hydrochloride. whakaurua hoki i roto i tenei rongoā ngā wāhanga ngaahi houalotú pērā i anhydrous colloidal takawai, monohydrate reihuka, te konutai māngaro glycolate, stearate konupora me te MCC.

papa Kikī i roto i mōkihi namunamu me kātene aua.

Drug "Velaksin" - capsules, tohutohu hoki te whakamahi i E kopakia ana i roto i te tākai, pepa, gelatin me te mārō. E ratou pōtae karaka-parauri, me te tïpako taekore. Ko hoki te wāhanga kaha o tenei puka te venlafaxine pūhui. I tua atu ki tona hanganga o tenei rongoā ngā kai atu.

Ka rite ki nga mahi tarukino?

"Velaksin" - he whakatupuranga hou o anti-depressant. E ai ki te hanganga matū o tona taonga kaha e kore e no ki tetahi piha mohiotia o pōuritanga (hei tauira, tricyclic, tetracyclic, atu ranei). Tohunga mea e te tarukino he kaha enantiomer 2 racemate.

pā ana te parau tumu o te mahi o tenei tarukino te ki tona kaha ki te potentiate te CNS karere hihiko te tuku.

E ai ki nga tohutohu, venlafaxine me tona metabolite matua (EFA ranei e-desmetilvenlafaksin) tohu inhibitors puai o te reuptake o norepinephrine me serotonin me inhibitors ngoikore o te dopamine reuptake. E kore e taea e tatou te mea e, teie mau matū e taea ki te whakaiti i te mahi beta-adrenergic i muri i te rongoā kotahi, me te tamau. He rite whai hua ki reuptake o neurotransmitters EFA me venlafaxine.

He aha atu he tarukino faahiahia "Velaksin"? pūrongo Guide e te whakauru kaha o te tarukino he hunaonga ki a te mau farii ohipa N- me m-cholinergic, roro α1-adrenoceptors me histamine H1-receptors. I tua atu, inhibits reira te mahi o Mao me e kore faitatau ki fentsiklidinovymi, opioid, benzodiazepine me NMDA-receptors.

Ko te kinetics o te tarukino

ahakoa horomia te tarukino te, "Velaksin" (papa)? kī Tohutohu mō te Whakamahi e te tino pai whenumi te wāhanga hohe o tenei tarukino i te punuatuna. I muri i te horopeta kotahi o te medicament i roto i te inenga o 25-150 mg o tona kukū rawa i roto i te toto tae te i muri i 2.4 haora. Ko te kupu venlafaxine te ngā metabolized i roto i te haere tuatahi i roto i te ate. Ki te tangohia te tarukino i te kai, i te ona kukū piki tihi e 27-30 meneti i roto i te wē.

whakaaro te metabolite matua te he te tikanga o te e-desmetilvenlafaksin. Ko tōna hawhe-te ora me te whakakorenga hawhe-ora o te venlafaxine he 11 me te 5 haora, aua (putanga i roto i te puka tonu i nga whatukuhu).

Ko te kinetics o raau taero i roto i te āhuatanga haumanu motuhake

hiahiatia Drug "Velaksin" ako te pānui i roto i te iwi ki te cirrhosis o te ate he atu āhuatanga nekeneke. toto kukū o te raau taero nui haere i roto i enei tūroro, me tona tere o te papī, i runga i te anga ke, iti.

I roto i te kino iti hoki tākihi, täkihi me te āhua whakawātea katoa iti EFA me venlafaxine te ka roa te whakakorenga wā hawhe-ora te.

Me mahara hoki käore te reira e kore e te ira tangata me te tau o te manawanui pā te pharmacokinetics o te tarukino i raro i whakaarohia.

Tuhinga hoki

Aha tatou e hinaaro ai i te taputapu pērā i "Velaksin"? Ko te whakamahi o tenei tarukino whakaaturia i roto i te whārua o ngā takenga (mo te maimoatanga me te prophylaxis).

Ūhia ki te whakarite

I raro i te mea e kore e taea e tikanga te whakamahi i te tarukino "Velaksin"? Reviews o tūroro me kaiwhakaako titau e contraindicated tenei tarukino te ki riro:

  • i te fariiraa i Mao inhibitors ;
  • i roto i disorders tākihi nui;
  • i roto i te hapū whakapae whakapumautia ranei;
  • i roto i disorders nui o te ate;
  • i roto i te whāngai ū;
  • i roto i te taiohitanga me tamarikitanga, e ko, tae noa ki te tau o te nuinga;
  • ki te tūtohutanga tiketike ki te tarukino.

I tua atu, kia āta tangohia tenei tarukino i roto i angina iu, nui haere infarction myocardial (tae atu i te hou heke), takawhita, hītori haehae, tachycardia, mate taimaha, pēhanga intraocular, koki-katinga papahewa, predisposition ki toto i mucous me kiri, āhua härukiruki.

Drug "Velaksin" (papa): tohutohu mō te whakamahi

Raau "Velaksin" anake kia tangohia i roto i te kai. Ko te horopeta tīmatanga tūtohutia o te tarukino ko 75 mg, wehea i roto i te 2 werohanga wehea (i.e., 37.5 mg rua he ra), i tenei ra.

Ki te i muri i te maha o ngā wiki o therapy, e kore kua huru o te manawanui ake, kua nui haere te horopeta rā ki te 150 mg te ra, i roto i rua pota wehea (i.e., 75 mg rua he ra).

Ki te titau te manawanui he horopeta teitei o te raau (hei tauira, nui whakararuraru fakalotofo'í, ranei te tahi atu tikanga tono therapy pahoho), ka taea te kaitoi tautapa 150 mg o tarukino i roto i te 2 haora, a ka āta whakanui i te horopeta e 75 mg (2-3 ra i muri mai) ki te whakatutuki i te hua e hiahiatia ana.

E ai ki nga tohutohu, te inenga mōrahi "Velaksina" ko 375 mg ia ra. I muri te whakatutuki i te pānga e hiahiatia, e taea te āta tuku iho reira ki te taumata iti.

ārai matahoki me te tiaki therapy

tiaki tautoko o nga moni e taea te tango i te ono marama. I roto i tenei take, te rongoā tangohia i roto i te pota iti.

I roto i te iti hoki tākihi ngawari hiahiatia ako dosing talena te. I roto i te mate rite tūtohutia raro horopeta āhua i te 25-50%. Me mahara hoki käore te reira e kore e tika kia whakamahia venlafaxine i roto i nui iti hoki tākihi, mai kore ngā mōhiohio i runga i te haumaru o taua therapy ki te rā, e kore.

Iwi e te hunga i runga i tātari toto, kia riro 50% o te inenga mua rā o te raau taero i muri i nga pito wātū.

Hoki ngawari iti hoki te ako dosing talena ate kore hoki te hiahiatia. A, no te te mate, ko te kia heke horopeta āhua i te 50%. Ki te whakaaro ki kino kore ate, i roto i tenei take rāhuitia te whakamahi o te venlafaxine te.

I roto i te paari, kia whakamahia te tarukino "Velaksin" ki te tūpato tino. Ko e tika ana ki te tūkino taea o nga whatukuhu tenei. Me whakahau te tūroro i te horopeta whai hua i raro. I roto i tenei take, kia waiho te manawanui i raro i te tirotiro tamau hauora.

Whakakore raau

Runga ki te whakaotinga o te fariiraa i te tarukino kia whakaaro ki te whakaiti i te horopeta āta (i roto i te wiki). Kei te hiahiatia te reira ki te mau i te huru o te manawanui, i roto i te tikanga ki te whakaiti i te tūponotanga o tauhohe kino e pā ana ki te whakakāhoretanga o te tarukino.

Ko te wa e hiahiatia ana mo te mutunga oti o te rongoā, tei runga i te inenga, roanga o te therapy me takitahi ki takitahi.

pānga taha

He aha e nga pānga e hiahiatia o te tarukino e taea meinga "Velaksin"? Mua mea e te whanaketanga o te hunga ranei era atu meatanga kino e whai ake nei i te whakamahi o tenei taputapu, tei runga i te horopeta riro.

Ko te tauhohe tino auau te whakakitenga mai āhua tōraro ngā te whai ake:

  • takawhita, heke hiahia, moe rerekē, kōroke, ohoroa, whakapairuaki, Makere o, tremors, ruaki, cramps uaua, mangai maroke te kiri;
  • moemoea, kakā, mate taimaha, tachycardia, hyponatremia, tau'a, hypotension postural, whanoke, tauhohenga härukiruki, excitability manavasii, puare noa, paresthesia, syndrome neuroleptic, hiamoe, syndrome serotonergic;
  • nui haere oro uaua, hukihuki, dysuria, photosensitivity, te pupuri mimi, anorgasmia;
  • toto i roto i te kiri, ejaculation rerekē, menorrhagia, heke libido, sweating;
  • thrombocytopenia, raruraru noho, erythema multiforme, mydriasis, Stevens - Johnson, raruraru ataata, reka waimaero, Tuhinga o wa, ngoikore, ponana kiri, rohirohi, toto tauhohe anaphylactic.

Me mahara hoki käore te reira e muri i te withdrawal ohorere o te moni te whakaiti o tona inenga ranei e taea ngā pānga taha rite kārangirangi manavasii, rohirohi, korere, te momoe, tahurihuri kau, ānini, paresthesia, whakapairuaki, hypomania, ruaki, sweating, anorexia, ohoroa, maroke mangai, manukanuka, whanoke me te disorientation. Tikanga, He ngawari enei tohu, me te haere atu, kahore tetahi maimoatanga.

tūtohutanga

Hokona ahakoa pōuritanga kahore te whakahaunga? e kore he tino nui te rārangi o enei rongoa ( "Prozac", "Paxil", "Despres", "Azafen", "Pahi", "amitriptyline"), me te tarukino "Velaksin" Kei te kore ngā i roto i reira. E hoko i te reira i roto i pharmacies, taea e koe anake i te whakahaunga o te tākuta.

I mua i te tango i tēnei rongoā i raro i te arotake, rawa tūroro ki disorders fakalotofo'í, kia whakaaro te tūponotanga nui o ngā nganatanga suicidal. I roto i tenei whakaaro, i te timatanga o te therapy tarukino tūtohutia hoki te whakamahi i roto i te horopeta iti me i raro i tata te tirotiro hauora.

Iwi ki disorders huru i roto i te maimoatanga ki pōuritanga kia whakawhanake āhua härukiruki hypomanic ranei.

kia tino ki te whakatupato o te hiahia ki te kite i tonu he tākuta i te take o ngā huānga urticaria, rashes mate pāwera ranei tūroro.

Ētahi tūroro i roto i te tukanga o te fariiraa i venlafaxine kitea he hua horopeta-ti'aturi i roto i te pēhanga toto.

kia whakatupato tūroro ruhiruhia o te ofatiraa taea o te tikanga o te pauna, me te whanoke whanaketanga.

I roto i te maimoatanga o te moni kia karo tango inu waipiro.

Raau "Velaksin": mua manawanui, analogues hua

He aha te iwi e mea e pā ana ki tenei tarukino ki te manawanui? Kua korerotia maha kiritaki he maha nui o ngā pānga taha e puta i te tango i tēnei rongoā. Tino maha tenei tarukino ai tauhohe kino pērā i te momoe, ngoikore, ohoroa, hukihuki, whakaaro rerekē, whārua me te whakama. I tua atu, titau te tahi mau tūroro e noho enei pānga i muri i te otinga o te maimoatanga. Ano, he maha ngā kaiwhakamahi amuamu e pā ana ki te ahua o tohu withdrawal , me te ti'aturiraa.

He aha e taea e whakakapi raau pērā i "Velaksin"? Kei te kore ki te e kitea Analogs o tenei tarukino i roto i drugstores katoa. Ka rite ki te tikanga, ngā tohunga enei te whai ake: "Venlafaxine Sandoz", "Efevelon", "Alvent", "Nyuvelong", "Velafaks", "Dapfiks", "Voksemel", "Venlaksor", "Vensuert", "venlafaxine".

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