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Tohutohu mō te whakamahi "tiapridal". Analogs me arotake

"Tiapridal" - te rongoā whakakore hangaia e tiapride. tono te raau e rite te whakarokiroki, analgesic me hypnotic. Pūtake o te mahi ähotea - ārai i te mau farii ohipa dopamine, e tino pā te mahi o te CNS. I roto i tēnei tuhinga whakaahua tatou i roto i ngā kōrero e pā ana ki te tarukino.

Composition ngā te tarukino

E wātea ana i roto i te puka e rua, e taea te hokona te papa me te otinga te rongoā:

  • Kotahi papa rite kotahi ampoule Kei 100 milligrams o te wāhanga matua, me te matū pŭpŭ tauturu. Ka rite ki te kai mau pŭpŭ tauturu whakamahia i roto i te hanganga o te povidone, konupora stearate, mannitol. Kei te kō atu hoki te hanganga ki te hāorarua colloidal, silicon me te microcrystalline cellulose wai.
  • I tua atu i te wāhanga matua o te otinga Kei roto konutai pūhaumāota me te wai mo te werohia.

I roto i te pouaka kotahi roto 20 papa (2 opupu ki 10 papa) ranei 12 oko (2 opupu o 6 oko). Tohutohu mō te whakamahi "Tiapridal" i roto i te puka o te otinga mō te werohia taea whakahaerea e pâmuhia me intramuscularly. he pai anake hoki te maimoatanga o te tūroro pakeke tenei ahua o te tarukino.

Pharmacodynamics "tiapridal"

Ko te medicament he neuroleptic, analgesic me te mahi anxiolytic. Ka rite ki te ā-ako, "Tiapridal" tīpakongia poraka te mahi o te D 2 receptors o dopamine pokapū. Ko te kupu i runga i D 1 receptors e kore pānga. Te raau whakakahoretia tangata o psoriasis, ina whakamahia i roto i te paari whakapiki i whakaaro.

Pharmacokinetics "tiapridal"

kitea whakahaere Intramuscular o te tarukino (200 mg) o tona taumata mōrahi i roto i te tinana kei muri i te 30 meneti, te whakamahi i te papa i te horopeta kotahi - 60 meneti. nui haere te bioavailability o te tarukino, i te whakamahia tonu i te aroaro o te kai ki 75% ki te 95%. No te mea taero taua piki whakamahi me tona taumata mōrahi i roto i te rauropi (40%).

Absorption i roto i te tinana, ko te pōturi i roto i tūroro paari. "Tiapridal" tohutohu mō te whakamahi pā ana ki te kaihoko whiti te placental me toto-roro tauārai. Kei te mohiotia te reira e i roto i te maimoatanga he reira i roto i te hanganga o te waiu, uma te tarukino. I roto i nga wahine, i te tango wāhanga o te tarukino tere atu i taua o te tangata (i runga i 2.9 haora), te rerekētanga ko te 0.7 haora. Pākia āhuatanga rite āhua. Ko te wahi matua o te tarukino (70%) nekehia te i te tinana i te whatukuhu tonu.

Tuhinga "Tiapridal" teuteu

Hei whakatinana i te therapy ki taero "Tiapridal" pānui e whai ake:

  • dyskinesia (tardive, māhorahora);
  • Gilles de la Tourette syndrome;
  • chorea;
  • disorders whanonga (pukuriri kāwanatanga, rōpū, et al.), hua i roto i te rere nui o te waipiro ma'i me tūroro paari;
  • faaiteraa kino i roto i te whanonga, pērā i kaitaua kāwanatanga me te rōpū;
  • mamae pūāhua tino (puka ma'i).

Contraindications, ki taotiaraa riro "Tiapridal" tarukino

Opani te whakapanga o "Tiapridal" tohutohu mō te whakamahi mō ngā tamariki nei tau he iti iho i te ono tau. I roto i te therapy pediatric kawea i roto pire anake. E kore e te tarukino kia tukinotia hapu wahine me tūroro e whāngai ū. e kore te rongoā e whakamahia ana i roto i te take o te hypersensitivity ki ona wāhanga, me ētahi atu tikanga pera. Contraindications ngā taua āhua:

  • ate me te mate täkihi, e kua nui pakeke;
  • prolaktinzavisimogo Tātarihia te pukupuku, māharahara o tona aroaro;
  • raruraru hypertensive;
  • tātaritanga o te pheochromocytoma, he māharahara o tona oraraa.

Papa me te otinga whakamahia te tahi ki "sultopride" me agonists dopamine receptor (te okotahi ko te maimoatanga o te tūroro ki te mate o Parkinson) e kore e ngā ki etahi momo o neuroleptics, māngai anti-arrhythmic no ki ngā akomanga e ahau ko III A.

e kore e tukua Medicating "Tiapridal" ako wā kotahi te whakamahi i "Moxifloxacin", "sparfloxacin", "Difemanila", "erythromycin", "bepridil," "mizolastine", "levodopa", "cisapride" me ki rō-uaua "vincamine" .

Ki te te tukinotia te manawanui (ina koa te paari) ki taero e kia arahi ki te whanaketanga o te hypokalemia, ino āriponga cardiac, tawharara wā QT, te takanga o te bradycardia faaite huru, te whakamahi i te "Tiapridal" kia āta. hiahiatia tūpato te i roto i ngā take pēnei i:

  • mate o Parkinson;
  • congenital QT pūāhua elongation wā;
  • hypokalemia;
  • täkihi ma'i;
  • bradycardia;
  • mate i roto i i raru te pūnaha Cardiovascular (decompensation taahiraa);
  • haurangi.

Maimoatanga ki "Tiapridal"

i runga i te tono o "Tiapridal" ā taunaki te whakamahi i te tuatahi i roto i pota iti, āta piki haere ratou, i roto i te tikanga ki te whiwhi i te pānga mōrahi.

disorders whanonga

he tika hoki ratou te tauturu ki te tono 200 mg o te tarukino rā (ki runga, ki te 300). tutuki ana te pānga pai i roto i te ono wiki i runga i toharite. tūroro pakeke whakahaere he horopeta raro o te rongoā - 50 mg. kia pau te horopeta kotahi rua he ra, a ka tukua ona hua e i roto i te hanganga ture ki te wā whakapūtā, whakamana te mahi kei te āta, tango ki tohutohu tohunga pūkete. E kore e te horopeta rā nui 300 mg.

mamae kaha ma'i

Ko te horopeta rā o te tarukino mo te maimoatanga o taua tikanga he i 200 ki te 400 mg.

Chorea, Gilles de la Tourette syndrome

A, no te mau ana i roto i te maimoatanga o te tamaiti horopeta rā tīpakohia te tango ki te pūkete te taimaha tinana, me te pā ana ki 3-6 mg / kg. Ki te hiahia koe ki te whakahaere i te therapy pakeke, whakamahia tuatahi 25 mg o te raau taero ia ra, i muri mai (i muri i te hua āta i roto i te horopeta) - 300-800 mg.

Rōpū, fakaaoao

Ko te horopeta tūtohutia rā o medicament ko i 100 ki te 150 mg.

disorders whanonga

Ko te horopeta tūtohutia hoki te whakamahi awatea (i 200 ki te 300 mg) i roto i te take o āhua kuawa predelirioznogo ranei te putanga mai ki te 400-1200 mg. Ko te horopeta taea mōrahi e kore te tikanga e nui, ko te 1800 mg. Ko te kupu whakataki o te tarukino whakaputaina i runga i toharite katoa e rima haora. Ki te he tika hoki te tangata ruhiruhia maimoatanga, i nga ra katoa he 2-3 werohanga i waenganui i ai kite wā o 6 haora. Hoki te maimoatanga o taua tūroro rōpū rā, o 200 ki te 300 mg o medicament i whakaaetia te wa e ki te tomo iti iho i te 100 mg "tiapridal" tūtohutia.

faaiteraa Kakati o te āhua ma'i o te mamae

Whakaora i runga i te horopeta whakahaere rā e ōrite ana ki te 200-400 mg o te tarukino.

pānga te taha, no te tango "Tiapridal" tarukino

A, no te penei ā-tarukino "Tiapridal" ako, whakau arotake te tūponotanga o etahi tauhohe kino. kia puta Tūkinotanga i te urogenital, io, endocrine me ngā pūnaha Cardiovascular. I tua atu, i reira he he mōrea o ngā raruraru ki te rongo. Hoki ētahi atu pānga kino ngā mate pāwera, tahi faaiteraa kiri i taonga taimaha, hypotension orthostatic.

Tuwhena rawa "tiapridal"

Ki te whakamahi koe i horopeta nui tuwhena rawa taea, me ona tohu ngā raruraru o te mahara, te nui te nuinga o nei - pōroa, syndrome neuroleptic (mārere, ngā whakapeka). I roto i te tikanga ki te whakatika i tenei āhua o te kaiao kawea i roto maimoatanga e hāngai ana i runga i āpiha anticholinergic. I muri i te whakakāhoretanga o te tika tarukino ki te kawe i roto i te maimoatanga symptomatic me plasmapheresis.

Ara

I mua i te whakamahi taunaki ana te rongoā "Tiapridal" ā-ako e fakatonutonu koe hypokalemia. I roto i therapy he mea nui ki te aroturuki tonu kawehiko toenga, whakahaere he hiko-, aroturuki i te huringa pikitia haumanu.

Ki te mea e tika ana ki te tono hua te fariiraa i neuroleptics syndrome extrapyramidal whakawhanakehia hei utu o dopamine receptor agonist taero anticholinergic.

I te wa o te maimoatanga e whakarere ngā mahi e tū he riri pea, e kore e tūtohu ana ki te mahi i te mahi tono tiaki motuhake, me te whakautu tere.

Ngā pāhekoheko ki ētahi atu matū

Ētahi taka i ngā ki te tango rongoā "Tiapridal" ako, urupare e pā ana ki te tūponotanga o te takanga o tauhohe koretake te. E kore e tūtohu ana i roto i te maimoatanga tono "Clonidine", antihistamines, anxiolytics, barbiturates me opioids, rite ka waiho atu korerotia "tiapridal" pānga. Nā ki te incompatibility kore e tangohia "levodopa" me te waipiro. Ka taea te ngā rongoā ki te whakamahi o neurotrophic taero, Pë, pōuritanga, neuroleptics. mōrea tiketike o hypotension orthostatic, i reira ko te whakamahi tukutahi o raau taero antihypertensive ki "Tiapridalom".

Ko te utu o analogues tarukino, arotake e pā ana ki te tarukino "Tiapridal"

Ki te maimoatanga tika "Tiapridal" tikanga whakaahuatanga ako kia mohio koe ki ta te tarukino ko. He o faufaa nui i roto i te kōwhiringa o te medicament mo te maimoatanga i te utu o te raau taero. Ko te otinga i roto i te oko e taea te hokona hoki e pā ana ki 995 moni, me papa - no te 1,400 moni.

I roto i nga analogues o te tarukino - "Eglonil", "Betamax". O te whakakapi kia kia tīpakohia "Sulpiride" ranei "Prosulpin". He ko tetahi orotahi o te tarukino - "tiaprid", e whakaaro ia te tino wātea, ko reira tino he kōwhiringa rongonui, te hanga tarukino motu e ni'ai te kamupene "Organic". Hei wāhanga o "tiaprid" tapae te taonga kaha taua, e ko wāhanga o te rongoā "Tiapridal". E taunaki ana analogs Raihana Guide ki tīpako, ka kore e taea te whakamahi i te taketake tukutahi ki etahi taero ai ngā pānga taha me e kore e whakarato i te pānga e hiahiatia ana. Ki he whai hua te nuinga te raau taero, tango ki tokomaha o nga ngā pūkete ka tīpakohia.

I roto i te maimoatanga, he mea nui ki te whai i tohutohu katoa o te tākuta me ngā tūtohutanga, e kei tohutohu mō te whakamahi. "Tiapridal", rite whakaaturia e urupare, i nuinga o te wā, kei te whakamahia ki te whakakore i te tikanga haere tahi e te oaoa io me whanonga kaitaua, āhotea waipiro. Ko te tikanga, tūroro me ngā tākuta e makona ki te hua o te therapy. Fele, e kore te he akoranga whakahauora e hiahiatia ana mo te take e te whakawhanake i te pānga e hiahiatia ana i muri i te whakatinanatanga o te akoranga tuatahi. whakaatu Reviews i hoki tūroro rongoā "Tiapridal" ngāwari ki te whakamahi.

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