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Ko te tarukino "Sulpiride": arotake, tohu, analogs

Āhotea o rerekē te pakeke haere tahi tangata ake. Neke atu i te rau tau maha i whakapono ai e nohoia e te rewera i roto i te tangata mate, ka kua reira "rongoa" tenei raruraru kua tika. I mua ki te hanga o te manawa rongoā neuroleptic o disorders hinengaro whakaputaina maimoatanga otaota whakawhanakehia i runga i te pūtake o Belladonna, henbane, opiates. Mahi rite maimoatanga ki te konupūmā (rō-uaua), me te iriiri i te manawanui i roto i te tarukino moe.

Ka taea te huaina e te chlorpromazine ähotea rawa tuatahi, i mātātoa i whakamahia mo te maimoatanga o te tūroro ki te raruraru hauora hinengaro mai i 1953. I tēnei wā, ko te rārangi o rongoā mate ähotea, tino whakawhānui antipsychotics. Ko tētahi o raau taero whakamahia whānuitia o tenei rōpū ko "Sulpiride". Mua whakaahua ia rite te mate ähotea tino mohiotia.

pharmacodynamics o te tarukino

Neuroleptic pānga "sulpiride" antidofaminergicheskim e pā ana ki te mahi, m. E. I roto i te poraka tarukino pūnaha io pokapū nuinga receptors dopaminergic. Dopamine Ko te wāhanga nui o te "pūnaha utu" o te roro - whakaongaonga te sensation pai, makona atu, i roto i te tahuri, pānga te tukanga mātauranga, me te whakahihiko. I roto i te pota nui tiketike, whakaputaina i roto i te tukanga o tetahi wheako pai (i runga i te whakaaro tuakiri o te tangata) - fariiraa o te kai reka, he sex, kahore sensations tinana ahuareka. Ki te pai ake te nui te whakanui ake o dopamine i roto i te pūnaha io pokapū te whakamarie hinengaro, ki te hekenga - whakawhanake tohumate o te korekore.

Mahi "sulpiride" i rawa 600 mg (nui o rongoā ia) he horopeta ko te āhua mate ähotea. Ki te nga toketaá iti iho i te 600 mg - stimulant atu lahi me ngā pānga raau. Heoi serotonicheskie, histamine, adrenergic tarukino receptors he iti pānga.

Rongoā - analogues

Ko te medicament "Sulpiride" - neuroleptic mohiotia, no ki te rōpū o benzamides whakakapia - kua he maha makona nui o rongoā e he rite i roto i te hanganga me te he pānga. He taero e ōrite te waehere taumata ATC 4. Ko te "Betamax", "tiaprid", "Eglonil" enei. I tua atu i enei, he tono whanui kiritaki "Prosulpin", "Eglek" "rere" "Vero Sulpiride", "Sulpiride Belupo." Ka taea e whai Reviews o nga rongoa katoa e kiritaki e rua aronga pai, me te kino. Te reira i katoa tei runga i te pakeke o te kāwanatanga o hauora o te manawanui, tona te tūtohutanga ki te whakauru matua kaha - sulpiride, me te inenga o te tarukino whakaritea ki te farii i te tākuta.

Tuhinga ki te farii i rongoā

Sam neuroleptic "Sulpiride", ona analogs i te poi tika whanui o te mana, me te taea te whakaritea ki te farii i te mate makona nui. Tangohia te reira i roto i te aroaro o te wairua tuakoi i roto i nga wāhanga whakapeka, a ka he te reira ma'i. whakatikaia Sulpiridsoderzhaschih te whakamahi o antipsychotics i roto i te wā whakapeka o te whanaketanga o te kuawa (te mate hinengaro o te natura, haere tahi e te ngangau o te mahara mai i whanoke me te noa pōroa). Tino maha whakaritea te tarukino te mo te ngā disorders pōhewahewa me korekore, ahakoa o ratou take.

A, no te taninito o te take rerekē taunaki tango "Sulpiride" ā-ako. E pai te āhuatanga arotake o tūroro me kaimahi hauora medicament i roto i te rongoā neuritis vestibular, ka momo kore vertebrobasilar-basilar ki pāpāho otitis me traumas cranial, ki te mate o Meniere (nui haere rōrahi o te wai i roto i te kōhao taringa roto, e e pēhanga i runga i te pūtau mana ki te pupuri tauritenga te tinana me tona takotoranga i roto i te wāhi).

Ka rite ki te "Sulpiride" wahi o te therapy whānui taea te whakamahi i roto i ngā mahi haumanu mō te mate whewhe keté, me te syndrome whēkau pukukino.

Ko wai e pehi i tango taero ähotea i runga i te pūtake o te sulpiride?

Neuroleptics "Sulpiride" analogues tarukino o te whakauru matua kaha he rārangi motuhake o contraindications. Kaua e tangohia e te reira ki te iwi ki te hypersensitivity ki sulpiridu me te mamae i hyperprolactinemia (tino piki taumata o te prolactin taiki i roto i te toto). Fakatatau ki ai, e kore te tenei tarukino whakaritea ki te pukupuku prolactin-ti'aturi (mate pukupuku uma, prolactinoma repe , me ētahi atu).

I tua atu, "Sulpiride" (tohu whakaahuatia ana i runga) opani ako i roto i te pheochromocytoma (kaha hormonally pukupuku pūtau chromaffin), āhotea härukiruki me ngā disorders pängia ki haurangi fakaaoao whanonga. Kaua e whakamahi i tenei sulpiridsoderzhaschih rongoā ki te puipuitua o haurangi waipiro whakapeka, pau ki hypnotic taero rongoa me Pë whakapōauau.

E kore e whakaaturia Ko te whakamahi o te neuroleptic "Sulpiride" tūroro pakeke i raro i te 18 tau, me nga wahine i roto i te hohipera.

pānga taha pea o

tauhohe kino ki te neuroleptic ia me analogues "sulpiride" mua manawanui me ngaio hauora tohu rite feunga nui, tino ähua i te huru o te tūroro. He he he pea o te hyperprolactinemia i roto i te whānuitanga o ngā puka (gynecomastia, dysmenorrhea, frigidity, mananga iti, galactorrhea, hua i roto i te taimaha tinana).

Atu faaiteraa taea o te syndrome extrapyramidal, whakakitea nei e disorders pathological o te nui me te kounga o te kaupapa noa whakaputaina e uaua kōhiwi, te huri i roto i te reo uaua. Heoi, e kore te mea pāpāngia he tohumate e haapapu te meka o syndrome extrapyramidal.

Ka rite ki tauhohe taha ki "Sulpiride" analogs neuroleptic, kia puta faaati, akathisia (ngoikore ki te kia i te okiokinga), dyskinesia, ohoroa, te momoe, manukanuka excitability tiketike, te kārangirangi. Ka taea e whakaatu tohumate o syndrome mārere neuroleptic, āhuatanga e abnormalities autonomic, koma kiri, tūāhuruiti.

pānga te taha i te wahi gastrointestinal kia he sensation o maroke i roto i te mangai, te whanaketanga o te tokopā, whakapairuaki ahua, retching, kōroke. whakahohenga pea o transaminases ate, me te kawakore phosphatase.

tono pūnaha Cardiovascular "sulpiride" taea te whakautu i te hua i roto i te pēhanga toto (uaua - he hekenga i roto i te pēhanga toto, whanoke), nui haere auau ngakau, nui haere QT-wā. Tino uaua, engari ka taea e koe te whakarongo e i runga i te "Sulpiride" whakautu tarukino i rata tohu te momo o te arrhythmia torsadedepointes whanaketanga.

faaiteraa pāwera pērā i ponana kiri, pruritus, pāpaka eczematous. I te tahi taime e taea e koe te whakarongo e pā ana ki te takahi o te acuity ataata.

aratau dosing me te ara iahiko tono

E ai ki nga tohutohu mo te whakamahi o te medicament, tūroro nuinga pakeke i runga i te mate horopeta whakaritea o 100-300 mg ia ra rānei (wehea ki 2-3 werohanga). otinga waha e whakahaeretia ana i roto i te inenga rerekē: 100-800 mg ia ra mō te whakahaere intramuscular (i mua i te whakamahi tika ruru). Ko te mōrahi horopeta nohotahi hoki te pakeke, ko te 1.6 g

Ki te riro te reira e tika ana ki te tautapa "sulpiride" ki ngā tamariki i raro i te 18 tau o te tau, kia tātai i te inenga tango ki pūkete te taimaha i runga i te pūtake o te 5 mg ia manokaramu o taimaha tinana.

Ki te mea he huru o āhotea i roto i te wā whakapeka ma'i ranei te manawanui, therapy tikanga tīmata ki te whakahaere intramuscular (400-800 mg ia). I roto i te nuinga o te wā, te wā o te maimoatanga he i te iti rawa 2 wiki. Ka rite ki te hauora o te manawanui, i te werohia intramuscular whakawhitia ki te fariiraa "sulpiride" i roto i te pire. Neuroleptic "Sulpiride" arotake manawanui whakaahua hei rongoā whai hua. Ka taea te whakaritea roanga o te akoranga o te therapy, ka puta ke anake i te rata haere.

pota nui

Tetahi tohu motuhake e tohu ana i te meka o rawa nga pota whakaaetia mōrahi i runga, e kore. Ko te tikanga i roto i teie mau huru, i reira he pēhanga toto nui ake, kite te peroo. Pea te whanaketanga o te whakarokiroki (pehanga o te mahara i whakapataritari e taero, reka pānga, i pota teitei - hypnotic). I roto i te nuinga o te wā, nga pānga o te tarukino tohu "Sulpiride" mua manawanui te ahua o te whakapairuaki, mangai maroke, nui haere sweating, ruaki. I roto i te wā onge whakawhanake tohu extrapyramidal, Ka taea e gynecomastia puta tūroro tane (whakarahi uma). Tino uaua korero o parkinsonism korerotia, pōroa.

Ka rite ki raau whiriwhiri mō "sulpiride" tuimotu, e tūtohu maimoatanga symptomatic, i runga i te huru o te manawanui rānei. I roto i ētahi wā, te tono mahi pokapū holinoblokatory.

I te mea ki te whakarongo ki?

Tino hua katoa rōpū ähotea (tae atu sulpiridsoderzhatsie "Betamax", "Vero Sulpiride", "Prosulpin", "Sulperid Belupo", "Eglonil", "Sulpiride") arotake tohunga me tohutohu whakahaere, me te opani te papamuri o inu waipiro. tūtohutia hoki te tūroro ki te haurangi, ki te whakahaere rangahau haumanu, me te electrophysiological kua sulpiride Whakahekea reira te paepae mō te mahi ärai. Ki te whakamahia te tarukino te concomitantly ki taero e whakanui i te mōrearea o arrhythmias ventricular, taua tūroro titau aroturuki auau o te hiko-. Tei Nui ake QT-wā i runga i te horopeta.

Ki te i roto i te maimoatanga, i "sulpiride" tohu o tūāhuruiti (he meka e tohu ana ki te whanaketanga o te syndrome mārere neuroleptic), i te whakamahi o te tarukino kia mutu.

mutunga Inamata o therapy "sulpiride" taea whakapataritari tohumate withdrawal. Ko reira Maltitol i te raau hanga reira e taea ana ki te whakamahi i te iwi e mate ana i te huahuka ātete.

I roto i te wā maimoatanga katoa kia tūpato o waka me te whakatinanatanga o ngā mahi whakahaere tono whakamātau tinana whakautu tere, me te kukū tiketike.

rongoā Sulpiridsoderzhaschie me te hapū

Women i roto i te hapū "arotake Sulpiride 'mahue i roto i te ahunga tino pai. Mōrahi horopeta tīkina mō wahine hapu ko 200 mg ia ra kihai i whakapataritari pānga teratogenic (deflection o te whanaketanga embryonic). Ko te pota āhua nui o te tarukino mō wahine hapu No mōhiohio e wātea ana. Hoki, kahore he raraunga i runga i te pānga pea o taero-antipsychotics i runga i te whanaketanga roro o te tamaiti.

I roto i te whānui, e kore kaimahi hauora hiahia ki te whakamahi i "Sulpiride" mo te maimoatanga o wahine hapu, ki te kahore i roto i te wā i reira te pānga pai mō wahine kaha i runga i tūpono ki te kukune. I roto i ngā take pēnei i, "Sulpiride" ako (whakapumautia paramedics arotake) whakahaere taunaki i roto i te i raro pota ka taea, me te ki te taea ki te whakaiti i te wā o te maimoatanga.

I roto i te tamariki whanau ki te wahine tango i roto i rongoā sulpiridsoderzhaschie hapūtanga wā kite tohu gastrointestinal (bloating, a na i runga i. N.) Pāhono mana atropinopodobnye o neuroleptics. I te tahi taime e taea e koe te whakarongo e pā ana ki syndrome extrapyramidal. I roto i te whāngai ū mai "sulpiride" contraindicated.

Whakaaro o tūroro "sulpiride"

Ko te nuinga o nga tūroro i runga i te tarukino arotake "Sulpiride" rau te aronga pai. Neuroleptic makona whai hua, me te whakatika i te āhuatanga whakaaturia. Iwi tango "Sulpiride" ranei ona analogues mō tohu hinengaro i roto i whewhe pekitīlia whewhe duodenal ranei, korerotia te hekenga i roto i te kaha o te mamae puku, me te whakapai ake i roto i te huru whānui.

Kei te maha whakaritea pukapuka iti o te medicament (50 ki te 300 mg te ra) ki tūroro i tango i amuamu o whanoke auau puta hoki ngā take. I makona ki te hua o te maimoatanga te nuinga o enei tūroro.

pota nui "sulpiride" (neke atu i te 600 mg ia ra), i roto i te whakaaro o kaimahi rata ki te whakarato pānga ähotea whai hua i runga i ngā tūroro. Pota iti iho i te 600 mg, a i roto i te whakaaro o rata me tūroro, kawea whakaongaonga me te pānga raau.

He he he rōpū o tūroro e mahue te "sulpiride" i roto i te ara kino. whakawhanake e te mau taata whakapairuaki, oaoa, whanoke. ngaro tohu tōraro i muri korenga atu o te "sulpiride".

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