Hauora, Mau faaineineraa
Ko te tarukino "Captopril" i te aha? Taupānga, arotake, utu
He aha te te tarukino "Captopril", i nei te whakamahia reira me aha ngā āhuatanga? Ko te whakautu ki ēnei pātai katoa e taea e kitea i roto i te rauemi o tenei tuhinga. I tua atu, ka korero ki matou a koutou e pā ana ki te pehea, ki te tango i te tarukino me te aha ngā pānga taha me contraindications ki te whakamahi kua reira.
ngā mōhiohio whānui e pā ana te hua rongoa
Drug "Captopril" i roto i te reo Roma oro rite "Captopril". Tenei tarukino Ko te inhibitor waihanga o te whākōkī angiotensin-tahuri (ACE haapotohia ranei). Kei te whānui whakamahia ia i roto i te mahi hauora, ki tere whakaiti pēhanga toto.
Ko te hanganga, me te ahua o te tuku tarukino
Medicament "captopril" - i ai whakaritea te taputapu e ki? Tikanga, whakahau tākuta reira mo te hunga e mate ana e tonu i takawhita. raau Vauvauhia e hokona anake i roto i te puka o te papa spigot e kua whakanohoia i roto i te kātene. Ko te whakauru kaha o tenei tarukino ko captopril. Ko tōna ihirangi i roto i ia papa he 25 ranei 50 mg. kia kotahi mōkihi 100, 50, 40, 30, 20 ranei 10 nga wahi.
Ko te mahi pharmacological o te tarukino
Ka rite ki kōrero i runga ake, ki te ako "Captopril" papa ohanga e nei i roto i te kātene, ko te inhibitor o paru angiotensin-tahuri (ACE i.e.).
Me kï reira e e pā ana ngā āhuatanga antihypertensive o te tarukino me te inhibition whakataetae o mahi ACE, ārahi ki te faafariuraa auau heke nui o angiotensin 1 ki te angiotensin 2, i te mea he wāhanga vasoconstrictive tika puai.
I muri i te hekenga nui i roto i te kukū o te angiotensin 2 Ko te hua hia i roto i te wē mahi renin mā te whakakore i te urupare kino ina te tukua ai, me te whakaiti tika o te aldosterone production. I tua atu, i te medicament "Captopril", analogs nei e te aroaro ake nei, ka taea e whakaawe i te pūnaha kallikrein-kinin, ai te ārai i te rärangi o te bradykinin.
Nā ki te pānga vasodilating o te tarukino tino whakaiti te ātete katoa iaia (piringa), te pēhanga capillary poro me te pūkahukahu ātete iaia i roto i a ratou. I tua atu, he reira e taea ki te whakapiki ake i te rōrahi meneti o te uaua ngakau, me te faaohipa kātakí.
Ki te te tarukino "Captopril", arotake e pai ake o nei, te tango i te wa rawa te roa, ārai reira te whanaketanga o te kore ngakau, te whakaiti i te pakeke o te hypertrophy myocardial o te mānawanawa maui, me te pōturi iho te ahunga whakamua o te pū.
I tua atu, e taea ki te ārai i te ahunga whakamua o te nephropathy mate huka, e tukupu ana oro efferent arterioles tākihi, ka glomeruli tino whakapai ake hemodynamics intraglomerular te medicament ko.
Pharmacokinetics o te tarukino
I muri tango i te raau taero i roto ia hohoro whenumi. Ture haamata te medicament i muri e pā ana ki 40-60 meneti. tutuki ana te kukū mōrahi e i roto i te tinana tangata i muri i te haora tuatahi.
Me kï reira e te horomanga tukutahi o kai ki te tarukino hakari whakaiti i tona absorbability o 30-40%. Ko tenei he aha e tohutohu papa ki te tango i runga i 1 haora i mua i te kai i muri i 1-1.5 haora i muri ranei.
Roa o te mahi i muri i te whakamahi o te medicament (i roto i te tikanga ki te raro pēhanga toto), tei runga i te tini o tona fariiraa me te inenga. Hoki te whanaketanga o te pānga haumanu tonu kia rapua e te manawanui e rave rahi wiki o therapy.
Āhuatanga me ngā āhuatanga o te tarukino "Captopril"
Na e matau ana koutou e ko te tarukino "Captopril", Kei te whakamahia i ai reira me pehea ki te mahi i roto i te pā ana ki te tinana tangata. Ko ki matau te aha he pera rongonui tenei tarukino, kia whakaaro koe ona āhuatanga.
Ko te taonga kaha i te mea he wahi o "Captopril" teuteu roaa vasodilating, antihypertensive me āhuatanga cardioprotective.
Ko te ahei o te whakanui ake i te tuku o matū kaha biologically e whai he pānga natriuretic tenei tarukino. Nā ki tenei taonga tino whakapiki i rere toto ki nga whatukuhu. I tua atu, i te medicament "Captopril" o te pēhanga, me te whakaiti i te katoa pou-preload i runga i te ngakau, me piki i roto i te putanga cardiac.
Tuhinga hoki te whakamahi o te raau taero
tohua rongoā Vauvauhia mo te maimoatanga o te abnormalities e whai ake nei:
- takawhita matua me te renovascular. Ka taea te whakamahi i te reira i roto i ngā rite monotherapy ranei.
- Disorders o te mānawanawa maui. Tikanga, whakamahia te raau e ki aua iwi nei i te whakaeke ngakau, me te he inaianei i roto i te huru hauora pūmau.
- nephropathy mate huka. Tautapatia anake ki te hunga e he mate huka momo tuatahi, arā, te iwi taiāki-ti'aturi.
- Cardiomyopathy.
Drug "captopril" - i te mea atu te whakaritea tenei rongoa? Ka rite ki mohiotia te, e taea te aroaro te tarukino me te whakamahia i roto i te therapy matatini o te kore ngakau (congestive).
Contraindications ki te whakamahi o te medicament
E ai ki nga tohutohu, kei te tino riria te tarukino "Captopril" ki te tango i roto i te wā e whai ake nei:
- I roto i te take o te hypersensitivity ki te whakauru hohe - captopril. Me mahara hoki käore te reira e kore te tūtohu te tarukino mātātoa mo te hunga e whai he ātete i reira ko te mārama rōpū o taero, e he inhibitors o whākōkī angiotensin-tahuri (i.e., tūroro nei whakawhanakehia tetere angionefrotichesky i roto i te maimoatanga o te tahi atu inhibitor ACE).
- A, no te faaite mahi ate tangata.
- I roto i te ru cardiogenic.
- A, no te nga disorders kūnatu.
- A, no te whakahuatia tangata huru mahi tākihi i muri transplantation o te okana, stenosis më o pera, azotemia, hyperkalemia, me hyperaldosteronism tuatahi.
- Ki te hypotension.
- I roto i te mate immunological.
- stenosis Mitral me stenosis te pūtahi o.
I tua atu, e kore e te tarukino "Captopril" analogues o tenei tarukino tūtohutia hoki nga wahine hapu, tamariki i raro i te 18 tau o te tau, me te u.
Drug "Captopril": ako, te utu o te rongoā
E ai ki nga tohutohu piri, te tarukino kia e pā ana ki 1 haora tangohia i mua i ngā kai. kia tautuhia te roanga o te therapy me inenga talena o te rongoā te aroaro rata anake i runga i te pūtake takitahi, i runga i te momo, me te rere o te mate tīariari rānei.
Na me pehea ki te tango i te tarukino "Captopril"? Horopeta (tuatahi) o te medicament i te tātaritanga o te takawhita ko 12.5 mg rua he ra. I roto i te hiahia koi mō te kotahi wā e taea te whakamahi mo te faaineineraa o te 2 papa o 25 mg. Otiia i roto i tenei take, ko te minaminatia ki te kia wehea ki 3 ngā wā te fariiraa. Ko te horopeta mōrahi rā o te medicament taua he 150 mg.
Ki te mea kua whakaritea tō tākuta tiaki therapy mo te wa roa, te rongoā "Captopril", arotakehia matou tika i runga nei iteraa papû, kia tango i te papa tuatahi (25 mg) e toru nga wa ranei, e rua he ra.
A, no te takawhita renovascular me tākihi inenga tuatahi o te medicament ko 6.25 mg toru nga wa o te ra. Me uru therapy tautoko te waihanga 1 papa (25 mg) e toru ngā wā i te ra.
Ki te pāngia koe ki te kore te ngakau ma'i, me i reira he kōtītiti i nga whatukuhu, kia waiho te inenga tuatahi 12.5 ranei 6.25 mg toru nga wa o te ra. Ko te kupu kia kawea mai nga 2-3 wiki ki tona horopeta tiaki o 25-50 mg, me te auau taua. Ko te wā postinfarction tikanga tangohanga o medicament rite.
E whakaritea ACE rōpū o raau taero i roto i te paari ki te kaihaumanu anake. I roto i tenei take, kia wehewehea te maimoatanga. kia manakohia "Captopril" enei iwi te horopeta iti. I tua atu, e kore e tūtohu ana ki te whakapiki ake i puta noa te maimoatanga. A, no te tino tika, ato'a koe e taea te whakamahi i te diuretic koropiko.
Ko te utu, ka hoki 40 papa o tenei hua ka whai koe ki te utu e pā ana ki 50-60 moni Russian. Ka rite ki a koutou e taea te kite, te tikanga o "Captopril" Ko te tarukino āhua ngāwari e whai hua raro pēhanga toto i roto i te ara hauora.
Tangohia ki te tūpato tino
kia rongoā Vauvauhia kia tangohia ki te tūpato tino ka:
- inhibition o wheua wheua o te tohanga toto;
- nui mate autoimmune;
- mate huka;
- ischemia kaka ;
- mate ngakau coronary.
pānga taha
E ai ki nga tohutohu, i muri i te tarukino "Captopril" kia puta i roto i te tūroro e whai ake tauhohe taha:
- bronchospasm, Bronchitis, hāhā o te manawa, maroke mare huakore;
- CNS korekore, ānini, hukihuki, ataxia, whanoke, mania i nga topito o runga me raro, e rite ana te pai kia rite ki te mana'o o te kōpā, whakama, raruraru o kakara, me te kite, rohirohi, korekore;
- dermatitis exfoliative, minamina, ponana kiri, photodermatitis, pemphigus, angioedema, urticaria, ru anaphylactic, paitini necrolysis epidermal, alopecia;
- whakaoho manawataki ngakau, pectoris angina, hypotension orthostatic, infarction myocardial, tachycardia;
- reka ngangau, flatulence, mate o hiahia, stomatitis, whakapairuaki, kōroke, glossitis, pāpaka ulcerative o te mucosa pekitīlia me mangai, korere, ruaki, xerostomia, mamae puku;
- paresthesia, rumati, neuropathy piringa;
- neutropenia, hyperkalemia, thrombocytopenia, agranulocytosis, eosinophilia;
- oliguria, proteinuria, tākihi waimaero mahi;
- kakā cholestatic, pancreatitis, cholestasis, necrosis hepatocellular.
E ai ki ngā whakautu e waiho kiritaki o tenei tarukino, kia puta ngā pānga taha nui atu ki te, i te tango rongoā ki te ū ki iti-tote tote-free kai ranei.
Drug "Captopril": tuwhena rawa
I roto i te raraunga tuwhena rawa te tikanga e taea e tūroro faaite mai pānga taha pērā i infarction myocardial, ka whakahuatia e te maturuturunga iho tere i roto i te pēhanga toto, te ngangau i whakapeka o tohanga kaka me pōauautanga thromboembolic.
mehua whakatūpato
E ai ki te tohunga, e kore e tūtohu ana ki te tango i te tarukino me Diuretics pāhare pāporo-tohu, me ētahi atu taero e whakanui i tino te kukū o pāhare pāporo i roto i te wē toto. Ki te tau'a ore tatou i tenei Kaunihera, i reira te mea he mōrearea nui o hyperkalemia.
I tua atu, kia whakamahia tarukino "Captopril" ki tūpato tino ki fariiraa tukutahi tikanga "Procainamide", "" allopurinol "," Azathioprine "ranei te tahi atu immunosuppressants, rawa i roto i disorders o te mahi tākihi.
I roto i te E ruia ana mate kiko tūhonohono, me te kore ngakau ma'i, e titauhia anake te tarukino kia tangohia i raro i tata te tirotiro hauora.
Me mahara hoki käore te reira e, kia rite ki tūroro hauora me arotake, te pānga hypotensive o te medicament whakaiti tarukino "Indomethacin" me estrogens.
tikanga rokiroki
Drug "Captopril" e pā ana ki te B. Rārangi taero tukua tenei rongoā i roto i mekameka rongoā anake i runga i whakahaunga o tākuta. Ko tōna ora papa ko 3 tau i te rā o te whakanao. Taua tikanga Kei roto pai i roto i te wahi pouri, me te maroke, i te pāmahana e kore rawa 25 ° C.
analogues tarukino
E ai ki te whakauru kaha kua te analogs hanganga e whai ake nei o tenei tarukino:
- "Captopril Verein";
- "Angiopril-25";
- "Acre Captopril";
- "Alkadiene";
- "Captopril Sandoz";
- "Vero Captopril";
- "Captopril UBF";
- "Blokordil";
- "Captopril Akos";
- "Hexane Captopril";
- "Capoten";
- "Captopril FPO";
- "Captopril Sar";
- "Katopil";
- "Aegis Captopril";
- "Epsitron";
- "Captopril STI."
Ka rite ki te kite koe, rongoā tuku kua tino he torutoru ahurei. Na reira, tūroro maha whakaara ake te pātai o te mea te mea pai - te tarukino "Captopril" ranei "Capoten". Ko te rerekētanga tumuaki i waenganui ia ratou. rerekē ratou i ia atu anake e te kaiwhakanao. Hoki tenei take, te auraa "Capoten" he utu 3.5 wā atu te utu tarukino "Captopril".
Reviews o te faaineineraa
Ahakoa te utu iti, te medicament "Captopril" tōtika Whakahekea pēhanga toto. Tūroro e kua whakamahia toutou tenei tarukino mea e ona pānga kitea i roto i 1-3 haora i muri i ingestion.
Takitahi tauhohe mate pāwera i muri i tono o te kaihoko puta i roto i pā ana ki 5-8% o te iwi. He tokomaha tautohe e tenei raau ai tetere nui. Ko te aha i mua ki te whakamahi i, kia mohio ki te kōrero ki tō tākuta. Ki te nga tikanga o "Captopril" Ko te iti rawa kia kotahi pānga taha, he reira e minaminatia ki te paopao ki i reira, ka haere ki runga ki te rongoa mo te pēhanga toto tiketike i tetahi atu rōpū.
He he he rota tonu o arotake e "Captopril" taero "Capoten" me ētahi atu analogues o enei moni tōtika āwhina ki te pehea e o takawhita kaumātua. Otiia i mua i te tikanga taua, kia mohio ki te kōrero ki tō tākuta. I tua atu, ki te tangata i roto i te tau tawhito faaore pēhanga toto tiketike, me te tūtohu atu mate e ki te whakamahi i anake te horopeta i raro o te rongoā.
He mea haumaru ki te whakamahi i te tarukino?
I runga i te pūtake o te hōhipera ā-rohe i roto i Rivne (Ukraine) i roto i te 2010, i whakahaeretia he ako i auau o ngā pānga taha i tango i te tarukino "Captopril". I roto i tenei tukanga, tae e te iwi ki ngawari, me te āhua takawhita matua. Ka rite ki te hua, o nga kaupapa 500 amuamu o ngā pānga taha 73 anake te iwi. O enei, 53 - Kati tango i te raau taero, me te toe 20 - tonu, i kitea e ratou e hopoi mai te reira atu pai te rota atu kino ki te hauora.
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