Hauora, Mau faaineineraa
Buserelin taupuni - āhuatanga whakaahuatanga me te tono
kia hāngai te kōwhiringa o te tarukino hormonal i runga i te ako tupato o nga tohu, me te tāutu tupato o te mōrea o ngā pānga taha.
Te faaineineraa "Buserelin Depot" whakataurite pai ki ētahi atu o tona kakama tiketike, me te tūponotanga iti o ngā tohu kino. Ko ia he mema o āpiha anticancer hormonal.
Ko te mahi pharmacological o te tarukino
Kei te mahi o te buserelin antigonadotropnym, anti-androgenic, anti-estrogen, pānga anti-puku. Drug taonga "Buserelin Depot" i te whakataetae here ki receptors o ngā pūtau secreting take gonadotropin-tuku (e ratou i roto i te hanganga o te taupa mārōrō o te repe).
I roto i te wā tuatahi kitea te tāuru tarukino te he hua tūao i roto i te kukū o LH me FSH (taiki gonadotropic), tohaina e te rapae o, e tika ana ki te nui haere taihemahema ihirangi Gomonov. I muri i 14 - 21 ra ārai te tikanga mahi gonadotropic i feedbacks kino, e arata'i ki te whakaiti nui o LH ko FSH, a, rite ki te hua, me te hekenga i roto i te hanga o hormones sex. Ko te kupu, heke kukū testosterone tane, tae te reira i te taumata whakapumautia nei i muri i orchiectomy (castration hauora). tuku iho tarukino Women pānga "Buserelin Depot" te ki te taumata o te production estradioda ngā i roto i te wā posklimaktericheskom.
Whakamahi o te tarukino "Buserelin Depot"
Kei te whakamahia te reira i roto i te maimoatanga o te mate pukupuku repeure, i roto i ētahi wā, e whakamahia ana ki te pehi i te testosterone production i roto i te testes. whakamahia hoki i roto i te maimoatanga o te mate pukupuku uma (taiaki-ti'aturi mate, āhuatanga nei i te production teitei o estrogens ranei puta i roto i te endometriosis). Ētahi atu mate, penei "buserelina Depot": fibroids uterine, hyperplasia endometrial, whakahaere i te hōtaka IVF i roto i te rongoā te pākoko.
Contraindications me tūtohutanga motuhake
Hypersensitivity, orchiectomy, hapū, hohipera. Whakatūpatotanga tango te raau taero i roto i te māuiuitanga o te mimi i te taumata o te metastasis vertebral, takawhita, mate huka, me te whārua. Buserelin taupuni me te hapūtanga - ariā hotokore.
pānga taha
kia amuamu te manawanui o te ahuatanga i runga i te wahi o te pūnaha io pokapū i roto i te puka o pāhoahoa, pau te, ohoroa, mate wareware, heke kukū, whanoke, tapepe aronganui, a ētahi wā korekore. Ka taea te Ua ite te reira tinnitus pēhanga ranei i runga i te 'Afio, kite te peroo rongo ranei. Ka taea e maha e te reira "hiko wera." I roto i te wiki tuatahi o te maimoatanga i roto i nga wahine kitea psevdomenstruatsiya, ka whakaturia te maroke tara, ka taea wheua demineralization, heke libido. I roto i nga tangata, kia kino ake ngaa te mate i roto i te tuatahi 2 - 3 wiki, ranei puta gynecomastia, heke mananga. anorexia, disorders dyspeptic: tangohia kia puta taua. He hotokore Buserelin taupuni me te waipiro. I roto i te tūroro ki te takawhita kia whakanui i te pēhanga, auau ngakau. Mai i mate pāwera puta: minamina, hikaka, bronchospasm, ru anaphylactic. Te huri i tohu taiwhanga: dyslipidemia, Hyperglycemia, hua i roto i transaminases me bilirubin, thrombocytopenia me leukopenia.
Ko te mau parau tumu o te tarukino
whakahaere Intramuscular: whakahaere i muri tonu faaineineraa o te whakatārewatanga.
- ka repeure puku katoa 4 wiki i 4.2 mg.
- Endometriosis - kua whakaurua i roto i te 4 marama.
- ki te myoma -3 marama uterine.
- pākoko - 4.2 mg.
whakahaere Intranasal:
- mo te maimoatanga o mate wahine whakaahuatia i runga - whakahaere ki te kōhao nasal 900 mg / ra (kotahi horopeta, 3 ngā wā i te ra), i 1 - 2 ra o te huringa te paheketanga.
- pākoko 600 mg / ra, 1 horopeta i roto i te kōhao nasal wha nga wa ia ra. Ki te kaha te whakaputa pā o te pūnaha whakaputa uri, heke te horopeta e ki te 2 ngā wā.
Ētahi tuhipoka:
- kawea te rongoā o te matepukupuku repeure te puta noa te ora;
- drugs anti-androgen whakahaerea hoki 2 wiki. a mo te 2 wiki. o te maimoatanga me te buserelin, ārai pōauautanga e kia puta i roto i te wiki tuatahi o te maimoatanga;
- i roto i te wā tuatahi o te maimoatanga i roto i nga wahine kia kitea whēwhē ovarian;
- kia ārai hapū me te ārai te whiwhi rongoā ki te hamani buserelin, engari he tika ki te whakamahi i ngā tikanga kore-hormonal o te ārai te 2 marama tuatahi;
- te pānga pai i runga i te maimoatanga tarukino o endometriosis hāparapara i te whakaiti i te auau o relapses.
Ngā pāhekoheko ki ētahi atu taero
whakaiti Buserelin te pānga o raau taero hypoglycemic. kia meinga te reira i hyperstimulation ovarian, ki te whakamahia tahi me taero ngā hormones sex.
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